Lofepramine
Cat. No.:YN480790
产品名称: | Lofepramine |
CAS No.: | 23047-25-8 |
Chemical Name: | 1-(4-chlorophenyl)-2-[[3-(10,11-dihydro-5H-dibenz[b,f]azepin-5-yl)propyl]methylamino]-ethanone |
Synonyms: | Lopramine |
分子量: | 418.96 |
分子式: | C₂₆H₂₇ClN₂O |
SMILES: | CN(CC(C1=CC=C(Cl)C=C1)=O)CCCN2C3=CC=CC=C3CCC4=CC=CC=C42 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | Lofepramine (Lopramine) 是有效的三环抗抑郁药,广泛地代谢为 Desipramine。Lofepramine 的抗抑郁活性源于通过抑制摄取促进去甲肾上腺素能神经传递,并且还可以通过抑制神经元摄取 5-羟色胺和色氨酸吡咯酶来增强 5-羟色胺能神经传递。Lofepramine 除了具有抗抑郁作用外,还具有显着的抗焦虑功效。 |
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