ACT-389949
Cat. No.:YN480798
产品名称: | ACT-389949 |
CAS No.: | 1258417-54-7 |
Chemical Name: | |
Synonyms: | ACT389949,ACT 389949,ACT-389949 |
分子量: | 428.39 |
分子式: | C₂₀H₁₈F₂N₆O₃ |
SMILES: | O=C(C1=C(C2=CC=CC(C)=C2)OC(C)=N1)NC3=NN(CC4=NC(C(F)(F)C)=CO4)N=C3 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | ACT-389949 是一种首创、高效、选择性的甲酰肽受体 2/脂蛋白 A4 受体(FPR2)/(ALX)激动剂,对 FPR2/ALX 进行内化入单核细胞的EC50值为 3 nM。ACT-389949 具有研究炎性疾病的潜力。 |
IC50和靶点: | |
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In Vivo: | |
Clinical Trial: | |
Solvent & Solubility: |