AF64394
Cat. No.:YN480878
产品名称: | AF64394 |
CAS No.: | 1637300-25-4 |
Chemical Name: | N-[[4-chloro-2-(1-methylethoxy)phenyl]methyl]-5-phenyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine |
Synonyms: | AF64394;(4-Chloro-2-isopropoxy-benzyl)-(5-phenyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl)-amine;N-(4-chloro-2-isopropoxybenzyl)-5-phenyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine;BCP29864;AF 64394;AK00799739;N-[[4-Chloro-2-(1-methylethoxy)phenyl]methyl]-5-phen |
分子量: | 393.87 |
分子式: | C₂₁H₂₀ClN₅O |
SMILES: | ClC1=CC(OC(C)C)=C(CNC2=CC(C3=CC=CC=C3)=NC4=NC=NN42)C=C1 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | AF64394 是GPR3的逆向激动剂,其pIC50值为 7.3。 |
IC50和靶点: | |
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Jensen, T., Elster, L., Nielsen, S.M., et al.The identification of GPR3 inverse agonist AF64394; The first small molecule inhibitor of GPR3 receptor functionBioorg. Med. Chem. Lett.24(22),5195-5198(2014)