NF-56-EJ40
Cat. No.:YN480998
产品名称: | NF-56-EJ40 |
CAS No.: | 2380230-73-7 |
Chemical Name: | |
Synonyms: | |
分子量: | 443.54 |
分子式: | C₂₇H₂₉N₃O₃ |
SMILES: | O=C(NC1=C(CC(O)=O)C=CC=C1)C2=CC=CC(C3=CC=C(CN4CCN(C)CC4)C=C3)=C2 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | NF-56-EJ40 是一种有效,高亲和力和高度选择性的人SUCNR1 (GPR91)拮抗剂,IC50为 25 nM,Ki为 33.5 nM,对大鼠SUCNR1几乎没有活性。 NF-56-EJ40 对人源化大鼠SUCNR1具有高亲和力,Ki值为 17.4 nM。 |
IC50和靶点: | |
In Vitro: | |
In Vivo: | |
Clinical Trial: | |
Solvent & Solubility: |