S107
Cat. No.:YN481427
产品名称: | S107 |
CAS No.: | 927871-76-9 |
Chemical Name: | |
Synonyms: | S-107; S 10 |
分子量: | 209.31 |
分子式: | C₁₁H₁₅NOS |
SMILES: | COC1=CC=C2C(CN(C)CCS2)=C1 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | S107 是一种口服可用的,血脑屏障可渗透的化合物,通过增强 calstabin2 与突变 Ryr2-R2474S 通道的结合来稳定RyR2通道。S107 抑制肌浆网 (SR) 的 Ca2+渗漏,预防心律失常,提高癫痫发作阈值。 |
IC50和靶点: | |
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In Vivo: | |
Clinical Trial: | |
Solvent & Solubility: |