PD 404182
Cat. No.：YN481572
CAS No. ：72596-74-8
规格
价格(RMB)
库存
| 产品名称: | PD 404182 |
| CAS No.: | 72596-74-8 |
| Chemical Name: | 3,4-dihydro-2H,6H-pyrimido[1,2-c][1,3]benzothiazin-6-imine |
| Synonyms: | PD404182;PD-404182 |
| 分子量: | 217.29 |
| 分子式: | C₁₁H₁₁N₃S |
| SMILES: | N=C1SC2=CC=CC=C2C3=NCCCN13 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | PD 404182 是一种有效的、竞争性的人类二甲基精氨酸二甲基氨基水解酶 1(DDAH1)抑制剂，IC50值为 9 μM。PD 404182 在体外表现出抗血管生成和抗病毒活性。 |
| IC50和靶点: | |
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| Solvent & Solubility: |
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Kleinschek, A., Meyners, C., Digiorgio, E., et al.Potent and selective non-hydroxamate histone deacetylase 8 inhibitorsChemMedChem11(23),2598-2606(2016)
Birck, M.R., Holler, T.P., and Woodard, R.W.Identification of a slow tight-binding inhibitor of 3-deoxy-d-manno-octulosonic acid 8-phosphate synthaseJ. Am. Chem. Soc.122,9334-9335(2000)
