GAT228
Cat. No.:YN1710043
产品名称: | GAT228 |
CAS No.: | 1446648-15-2 |
Chemical Name: | 3-[(1R)-2-nitro-1-phenylethyl]-2-phenyl-1H-indole |
Synonyms: | GAT228; GAT-228; GAT 228; |
分子量: | 342.3906 |
分子式: | C22H18N2O2 |
SMILES: | O=[N+](C[C@H](C1=CC=CC=C1)C2=C(C3=CC=CC=C3)NC4=CC=CC=C42)[O-] |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | GAT228 是 GAT211 的对映体,是大麻素受体 1(CB1)的配体。 |
IC50和靶点: | |
In Vitro: | |
In Vivo: | |
Clinical Trial: | |
Solvent & Solubility: |
Laprairie, R.B., Kulkarni, P.M., Deschamps, J.R., et al.Enantiospecific allosteric modulation of cannabinoid 1 receptorACS Chem Biol.8(6),1188-1203(2017)
Mitjavila, J., Yin, D., Kulkarni, P.M., et al.Enantiomer-specific positive allosteric modulation of CB1 signaling in autaptic hippocampal neuronsPharmacol. Res.129,475-481(2018)