Methiothepin maleate
Cat. No.：YN1730142
| 产品名称: | Methiothepin maleate |
| CAS No.: | 19728-88-2 |
| Chemical Name: | 1-[10,11-dihydro-8-(methylthio)dibenzo[b,f]thiepin-10-yl]-4-methyl-piperazine, (2Z)-butenedioate |
| Synonyms: | Metitepine maleate; Ro-8-6837 maleate |
| 分子量: | 472.6222 |
| 分子式: | C20H24N2S2 • C4H4O4 |
| SMILES: | CN(CC1)CCN1C2C3=C(C=CC(SC)=C3)SC4=CC=CC=C4C2.OC(/C=C\C(O)=O)=O |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Methiothepin maleate 是一种有效的，非选择性的5-HT2receptor拮抗剂，pKd值为 7.10 (5-HT1A)，7.28 (5HT1B)，7.56 (5HT1C)，6.99 (5HT1D)，7.0 (5-HT5A)，7.8 (5-HT5B)，8.74 (5-HT6) 和 8.99 (5-HT7)，pKi值为 8.50 (5HT2A)，8.68 (5HT2B) 和 8.35 (5HT2C)。 |
| IC50和靶点: | |
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