Arformoterol tartrate
Cat. No.:YN1710048
产品名称: | Arformoterol tartrate |
CAS No.: | 200815-49-2 |
Chemical Name: | N-[2-hydroxy-5-[(1R)-1-hydroxy-2-[[(1R)-2-(4-methoxyphenyl)-1-methylethyl]amino]ethyl]phenyl]-formamide, (2R,3R)-2,3-dihydroxybutanedioate |
Synonyms: | 酒石酸福莫特罗; (R,R |
分子量: | 494.5 |
分子式: | C19H24N2O4 • C4H6O6 |
SMILES: | COC1=CC=C(C[C@@H](C)NC[C@H](O)C2=CC(NC=O)=C(O)C=C2)C=C1.OC([C@H](O)[C@@H](O)C(O)=O)=O |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | Arformoterol ((R,R)-Formoterol) tartrate 是 Formoterol 的 (R,R)-对映异构体,是一种长效 β2-肾上腺素能受体 (β2-AR) 激动剂,Kd为 2.9 nM。Arformoterol tartrate 可用于慢性阻塞性肺疾病 (COPD) 的研究。 |
IC50和靶点: | [{name:"Beta-2 adrenergic receptor:2.9 nM (Kd)"}] |
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Solvent & Solubility: |
Handley, D.A., Senanayake, C.H., Dutczak, W., et al.Biological actions of formoterol isomersPulm. Pharmacol. Ther.15(2),135-145(2002)