K-756
Cat. No.:YN310381
CAS No. :130017-40-2
产品名称: | K-756 |
CAS No.: | 130017-40-2 |
Chemical Name: | |
Synonyms: | K-756; K 756; K756; |
分子量: | 433.50 |
分子式: | C₂₄H₂₇N₅O₃ |
SMILES: | O=C1NC2=C(C=CC=C2)CN1CC3CCN(C4=C5C=C(OC)C(OC)=CC5=NC=N4)CC3 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | K-756 是一种直接的选择性tankyrase(TNKS) 抑制剂,抑制TNKS1和TNKS2的 ADP-核糖基化活性,IC50分别为 31 和 36 nM。 |
IC50和靶点: | [{name:"TNKS1:31 nM (IC50)"},{name: "TNKS2:36 nM (IC50)"}] |
In Vitro: | |
In Vivo: | |
Clinical Trial: | |
Solvent & Solubility: |