BQR-695
Cat. No.:YN420257
产品名称: | BQR-695 |
CAS No.: | 1513879-21-4 |
Chemical Name: | 2-[[7-(3,4-dimethoxyphenyl)-2-quinoxalinyl]amino]-N-methyl-acetamide |
Synonyms: | NVP-BQR695 |
分子量: | 352.39 |
分子式: | C₁₉H₂₀N₄O₃ |
SMILES: | COC(C(OC)=C1)=CC=C1C2=CC3=NC(NCC(NC)=O)=CN=C3C=C2 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | BQR-695 是一种PI4KIIIβ抑制剂,对于人类和疟原虫 PI4KIIIβ 的IC50值分别为 80 和 3.5 nM。 |
IC50和靶点: | [{name:"human PI4KIIIβ:80 nM (IC50)'}, 'Plasmodium', {'Plasmodium PI4KIIIβ:3.5 nM (IC50)"}] |
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McNamara, C.W., Lee, M.C., Lim, C.S., et al.Targeting Plasmodium phosphatidylinositol 4-kinase to eliminate malariaNature504(7479),248-253(2013)