Jaspamycin
Cat. No.：YN440146
CAS No. ：22242-96-2
规格
价格(RMB)
库存
| 产品名称: | Jaspamycin |
| CAS No.: | 22242-96-2 |
| Chemical Name: | |
| Synonyms: | 7-CN-7-C-Ino |
| 分子量: | 292.25 |
| 分子式: | C₁₂H₁₂N₄O₅ |
| SMILES: | O=C1C2=C(N([C@@H]3O[C@H](CO)[C@@H](O)[C@H]3O)C=C2C#N)N=CN1 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Jaspamycin (7-CN-7-C-Ino) 是一种有效的PKA激活剂，在Trypanosoma brucei中，与其 R 位点 (PKAR) 结合，EC50和Kd值分别为 6.5 nM 和 8 nM。Jaspamycin (7-CN-7-C-Ino) 不结合纯化的人 PKARIα。具有抗寄生虫活性。 |
| IC50和靶点: | [{name:"Trypanosoma brucei PKAR(199-499):6.5 nM (EC50)'}, 'Trypanosoma', {'Trypanosoma brucei PKA holoenzyme:8 nM (Kd)"}] |
| In Vitro: | |
| In Vivo: | |
| Clinical Trial: | |
| Solvent & Solubility: |
