PROTAC BET degrader-2
Cat. No.:YN430076
产品名称: | PROTAC BET degrader-2 |
CAS No.: | 2093388-33-9 |
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分子量: | 770.84 |
分子式: | C₄₁H₄₂N₁₀O₆ |
SMILES: | O=C(C1=NC(NC2=CC(C3CC3)=NN2CC)=C4C(NC5=C4C=C(OC)C(C6=C(C)ON=C6C)=C5)=N1)NCCCC7=CC=CC8=C7CN(C(CC9)C(NC9=O)=O)C8=O |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | PROTAC BET degrader-2 是一种强效的溴域及末端外 (BET)蛋白的降解剂,在 RS4;11 细胞中测得其对细胞生长的IC50值为 9.6 nM,并能实现肿瘤消退。 |
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