Tafenoquine
Cat. No.:YN250196
产品名称: | Tafenoquine |
CAS No.: | 106635-80-7 |
Chemical Name: | N4-[2,6-dimethoxy-4-methyl-5-[3-(trifluoromethyl)phenoxy]-8-quinolinyl]-1,4-pentanediamine |
Synonyms: | 他非诺喹; WR 238605 |
分子量: | 463.49 |
分子式: | C₂₄H₂₈F₃N₃O₃ |
SMILES: | CC1=CC(OC)=NC2=C1C(OC3=CC=CC(C(F)(F)F)=C3)=C(OC)C=C2NC(CCCN)C |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | Tafenoquine (WR 238605) 是一种 8-氨基喹啉。Tafenoquine 作为抗疟疾预防剂。 |
IC50和靶点: | |
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Coleman, R.E.Sporontocidal activity of the antimalarial WR-238605 against Plasmodium berghei ANKA in Anopheles stephensiAm. J. Trop. Med. Hyg.42(3),196-205(1990)
Marley, S.E., Eberhard, M.L., Steurer, F.J., et al.Evaluation of selected antiprotozoal drugs in the Babesia microti-hamster modelAntimicrob. Agents Chemother.41(1),91-94(1997)