Purfalcamine
Cat. No.:YN250262
CAS No. :1038620-68-6
产品名称: | Purfalcamine |
CAS No.: | 1038620-68-6 |
Chemical Name: | |
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分子量: | 528.62 |
分子式: | C₂₉H₃₃FN₈O |
SMILES: | O=C(C1=CC=C(NC2=C3N=CN(C4=CC=CC(F)=C4)C3=NC(N[C@H]5CC[C@H](N)CC5)=N2)C=C1)N6CCCCC6 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | Purfalcamine 是一种具有口服活性,选择性的恶性疟原虫钙依赖性蛋白激酶 1 (PfCDPK1) 抑制剂,IC50为 17 nM,EC50为 230 nM。Purfalcamine 具有抗疟疾活性,可以引起疟原虫在裂殖体阶段的发育停滞。 |
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