Nomegestrol
Cat. No.：YN480280
CAS No. ：58691-88-6
规格
价格(RMB)
库存
| 产品名称: | Nomegestrol |
| CAS No.: | 58691-88-6 |
| Chemical Name: | 17-hydroxy-6-methyl-19-norpregna-4,6-diene-3,20-dione |
| Synonyms: | |
| 分子量: | 328.45 |
| 分子式: | C₂₁H₂₈O₃ |
| SMILES: | C[C@@]12[C@](CC[C@]2(O)C(C)=O)([H])[C@@]3([H])[C@]([C@]4([H])C(C(C)=C3)=CC(CC4)=O)([H])CC1 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Nomegestrol 是一种有效的，可口服的孕酮，为选择性的孕酮受体 (progesterone receptor) 完全激动剂，对大鼠子宫孕酮受体的Kd值为 5.44 nM，具有很强的抗雌性激素活性，适度的抗雄性激素活性。 |
| IC50和靶点: | |
| In Vitro: | |
| In Vivo: | |
| Clinical Trial: | |
| Solvent & Solubility: |
Botella, J., Duc, I., Delansorne, R., et al.Structure-activity and structure-affinity relationships of 19-nor-progesterone derivatives in rat uterusJ. Endocrinol. Invest.13(11),905-910(1990)
