GSK963
Cat. No.:YN270045
CAS No. :2049868-46-2
产品名称: | GSK963 |
CAS No.: | 2049868-46-2 |
Chemical Name: | |
Synonyms: | GSK963 (Racemate) |
分子量: | 230.31 |
分子式: | C₁₄H₁₈N₂O |
SMILES: | CC(C)(C)C(N1N=CC[C@H]1C2=CC=CC=C2)=O |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | GSK963 是一种手性的、强效的、选择性的受体相互作用蛋白 1 (RIP1) 酶的抑制剂,其IC50值为 29 nM。GSK963 对体外小鼠和人细胞的坏死具有强效和选择性的抑制作用。 |
IC50和靶点: | |
In Vitro: | |
In Vivo: | |
Clinical Trial: | |
Solvent & Solubility: |