(+)-Norfenfluramine
Cat. No.:YN322810
产品名称: | (+)-Norfenfluramine |
CAS No.: | 19036-73-8 |
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分子量: | 暂无 |
分子式: | 暂无 |
SMILES: | 暂无 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | (+)-Norfenfluramine 是 (+)-fenfluramine 的主要肝脏代谢物,是一种选择性的5-HT2B受体激动剂 (Ki: 11.2 nM)。(+)-Norfenfluramine 有效地刺激磷酸肌醇的水解并增加细胞内 Ca2+。(+)-Norfenfluramine 可用于原发性肺动脉高压和心脏瓣膜病的研究。 |
IC50和靶点: | [{name:"5-HT2B Receptor:11.2 nM (Ki)"},{name: "5-HT2A Receptor:1516 nM (Ki)"},{name: "5-HT2C Receptor:324 nM (Ki)"}] |
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