CeMMEC1
Cat. No.：YN290105
CAS No. ：440662-09-9
| 产品名称: | CeMMEC1 |
| CAS No.: | 440662-09-9 |
| Chemical Name: | N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1,2-dihydro-2-methyl-1-oxo-4-isoquinolinecarboxamide |
| Synonyms: | CeMMEC1 HCl |
| 分子量: | 336.34 |
| 分子式: | C₁₉H₁₆N₂O₄ |
| SMILES: | O=C(C(C1=C2C=CC=C1)=CN(C)C2=O)NC3=CC=C(OCCO4)C4=C3 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | CeMMEC1 是BRD4的抑制剂，同时对TAF1有很高的亲和性，对 TAF1 的IC50值为 0.9 μM，对 TAF1 (2) 的Kd值为 1.8 μM。 |
| IC50和靶点: | |
| In Vitro: | |
| In Vivo: | |
| Clinical Trial: | |
| Solvent & Solubility: |
Sdelci, S., Lardeau, C.H., Tallant, C., et al.Mapping the chemical chromatin reactivation landscape identifies BRD4-TAF1 cross-talkNat. Chem. Biol.12(7),504-510(2016)
