Epertinib
Cat. No.：YN340062
CAS No. ：908305-13-5
| 产品名称: | Epertinib |
| CAS No.: | 908305-13-5 |
| Chemical Name: | |
| Synonyms: | S-22611 |
| 分子量: | 560.02 |
| 分子式: | C₃₀H₂₇ClFN₅O₃ |
| SMILES: | CC#C/C(C1=CC2=C(NC3=CC=C(OCC4=CC=CC(F)=C4)C(Cl)=C3)N=CN=C2C=C1)=N\OC[C@@H]5NCCOC5 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Epertinib (S-22261) 是一种有效，可口服，可逆的，选择性的EGFR，HER2和HER4抑制剂，IC50值分别为 1.48 nM，7.15 nM 和 2.49 nM。Epertinib 具有高效的抗肿瘤活性。 |
| IC50和靶点: | [{name:"EGFR:1.48 ± 0.0 nM (IC50)"},{name: "HER4:2.49 ± 0.1 nM (IC50)"},{name: "HER2:7.15 ± 0.5 nM (IC50)"}] |
| In Vitro: | |
| In Vivo: | |
| Clinical Trial: | |
| Solvent & Solubility: |
