(Rac)-Acolbifene
Cat. No.：YN481525
CAS No. ：151533-34-5
| 产品名称: | (Rac)-Acolbifene |
| CAS No.: | 151533-34-5 |
| Chemical Name: | 3-(4-Hydroxyphenyl)-4-methyl-2-[4-[2-(1-piperidinyl)ethoxy]phenyl]-2H-1-benzopyran-7-ol; EM 343 |
| Synonyms: | EM-343; (Rac)-EM-652 |
| 分子量: | 457.56 |
| 分子式: | C₂₉H₃₁NO₄ |
| SMILES: | OC1=CC=C2C(C)=C(C3=CC=C(O)C=C3)C(C4=CC=C(OCCN5CCCCC5)C=C4)OC2=C1 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | (Rac)-Acolbifene (EM-343; (Rac)-EM-652) 是 EM652 (estrogen receptor拮抗剂) 的外消旋形式，具有抗雌激素和雌激素活性。 (Rac)-Acolbifene (EM-343; (Rac)-EM-652) 含哌啶环，具有良好的药理作用，RBA=380。 |
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Gauthier, S., et al.: J. Enzyme Inhibition Med. Chem., 20, 165 (2005)
Tremblay, G., et al.: Cancer Res., 58, 877 (1998)
