Gestrinone
Cat. No.:YN480116
产品名称: | Gestrinone |
CAS No.: | 16320-04-0 |
Chemical Name: | 13-ethyl-17α-hydroxy-18,19-dinorpregna-4,9,11-trien-20-yn-3-one |
Synonyms: | 孕三烯酮; R 2323 |
分子量: | 308.41 |
分子式: | C₂₁H₂₄O₂ |
SMILES: | C#C[C@]1(O)CC[C@@]2([H])[C@]3([H])CCC4=CC(CCC4=C3C=C[C@]12CC)=O |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | Gestrinone (R 2323) 是一种合成类固醇激素,抑制平滑肌瘤的IC50值为 43.67 μM,有潜力用于子宫内膜异位症的研究。 |
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Moghissi, K.S.Medical treatment of endometriosisClin. Obstet. Gynecol.45(3),620-633(1999)
Tamaya, T., Fujimoto, J., Watanabe, Y., et al.Gestrinone (R2323) binding to steroid receptors in human uterine endometrial cytosolActa Obstet. Gynecol. Scand.65(5),439-441(1986)
Death, A.K., mcGrath, K.C.Y., Kazluskas, R., et al.Tetrahydrogestrinone is a potent androgen and progestinJ. Clin. Endocrinol. Metab.89(5),2498-2500(2004)