Giredestrant
Cat. No.:YN480413
产品名称: | Giredestrant |
CAS No.: | 1953133-47-5 |
Chemical Name: | |
Synonyms: | GDC-9545 |
分子量: | 522.55 |
分子式: | C₂₇H₃₁F₅N₄O |
SMILES: | OCC(F)(F)CN([C@@H]1C2=C(F)C=C(NC3CN(CCCF)C3)C=C2F)[C@H](C)CC4=C1NC5=C4C=CC=C5 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | Giredestrant (GDC-9545) 是一种非甾体雌激素受体 (ER) 配体,口服有效的,选择性ER拮抗剂。Giredestrant 可以在 ER 配体结合域内与雌二醇 (Estradiol) 竞争结合并诱导构象变化。Giredestrant 具有抗肿瘤活性。 |
IC50和靶点: | |
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Clinical Trial: | |
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