Enclomiphene citrate
Cat. No.:YN480695
产品名称: | Enclomiphene citrate |
CAS No.: | 7599-79-3 |
Chemical Name: | 2-[4-[(1E)-2-chloro-1,2-diphenylethenyl]phenoxy]-N,N-diethyl-ethanamine, 2-hydroxy-1,2,3-propanetricarboxylate |
Synonyms: | 恩氯米芬柠檬酸盐; (E)-Clomiphene citrate; trans-Clomiphene citrate; Enclomifene citrate |
分子量: | 598.08 |
分子式: | C₃₂H₃₆ClNO₈ |
SMILES: | Cl/C(C1=CC=CC=C1)=C(C2=CC=C(OCCN(CC)CC)C=C2)\C3=CC=CC=C3.O=C(CC(C(O)=O)(O)CC(O)=O)O.[(E)] |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | Enclomiphene citrate 是一种有效、可口服的oestrogen receptor拮抗剂,具有抗雌激素作用。 |
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Hill, S., Arutchelvam, V., and Quinton, R.Enclomiphene, an estrogen receptor antagonist for the treatment of testosterone deficiency in menIDrugs12(2),109-119(2009)
Wyss, R.H., Karsznia, R., Heinrichs, W.L., et al.Inhibition of uterine receptor binding of estradiol by anti-estrogens (clomiphene and CL-868)J. Clin. Endocrinol. Metab.28(12),1824-1828(1968)
Huang, S.-R., and Miller, W.L.Estrogenic and antiestrogenic effects of enclomiphene and zuclomiphene on gonadotropin secretion by ovine pituitary cells in cultureEndocrinology112(2),442-448(1983)
Weissenberg, R., Dar, Y., and Lunenfeld, B.The effect of clomiphene citrate and its Zu or En isomers on the reproductive system of the immature male ratAndrologia24(3),161-165(1992)