Raloxifene 4-Monomethyl Ether
Cat. No.:YN481237
产品名称: | Raloxifene 4-Monomethyl Ether |
CAS No.: | 185415-07-0 |
Chemical Name: | [6-Hydroxy-2-(4-methoxyphenyl)benzo[b]thien-3-yl][4-[2-(1-piperidinyl)ethoxy]phenyl]methanone |
Synonyms: | |
分子量: | 487.61 |
分子式: | C₂₉H₂₉NO₄S |
SMILES: | O=C(C1=C(C2=CC=C(OC)C=C2)SC3=CC(O)=CC=C31)C4=CC=C(OCCN5CCCCC5)C=C4 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | Raloxifene 4-Monomethyl Ether (Compound 37) 是一种 Raloxifene 衍生物,其抑制雌激素受体 α (estrogen receptor α)。Raloxifene 4-Monomethyl Ether 抑制 MCF-7 细胞,IC50为 1 μM,pIC50为 6。 |
IC50和靶点: | |
In Vitro: | |
In Vivo: | |
Clinical Trial: | |
Solvent & Solubility: |
Jone, C.D., et al.: J. Med. Chem., 27, 1057 (1984), Buelke-Sam, J., et al.: Reprod. Toxicol., 12, 217 (1998),