Raloxifene
Cat. No.:YN481353
产品名称: | Raloxifene |
CAS No.: | 84449-90-1 |
Chemical Name: | Keoxifene; LY 139481; [2-(4-Hydroxyphenyl)-6-hydroxybenzo[b]thien-3-yl][4-(2-(1-piperidinyl)ethoxy)phenyl]methanone; [6-Hydroxy-2-(4-hydroxyphenyl)benzo[b]thien-3-yl][4-[2-(1-piperidinyl)ethoxy]phenyl]-methanone |
Synonyms: | Keoxifene; LY156758 free base; LY139481 |
分子量: | 473.58 |
分子式: | C₂₈H₂₇NO₄S |
SMILES: | O=C(C1=C(C2=CC=C(O)C=C2)SC3=CC(O)=CC=C31)C4=CC=C(OCCN5CCCCC5)C=C4 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | Raloxifene (Keoxifene) 是一种苯并噻吩类选择性雌激素受体 (estrogen receptor) 调节剂 (SERM),对骨、血脂有雌激素激动作用,对乳腺和子宫有雌激素拮抗作用。Raloxifene 用于乳腺癌和骨质疏松症研究。 |
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Jone, C.D., et al.: J. Med. Chem., 27, 1057 (1984)
Buelke-Sam, J., et al.: Reprod. Toxicol., 12, 217 (1998)