Raloxifene hydrochloride
Cat. No.：YN481354
CAS No. ：82640-04-8
规格
价格(RMB)
库存
| 产品名称: | Raloxifene hydrochloride |
| CAS No.: | 82640-04-8 |
| Chemical Name: | [6-hydroxy-2-(4-hydroxyphenyl)benzo[b]thien-3-yl][4-[2-(1-piperidinyl)ethoxy]phenyl]-methanone, monohydrochloride |
| Synonyms: | 盐酸雷洛昔芬; Keoxifene hydrochloride; LY156758; LY139481 hydrochloride |
| 分子量: | 510.04 |
| 分子式: | C₂₈H₂₈ClNO₄S |
| SMILES: | O=C(C1=C(C2=CC=C(O)C=C2)SC3=CC(O)=CC=C31)C4=CC=C(OCCN5CCCCC5)C=C4.Cl |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Raloxifene hydrochloride (Keoxifene hydrochloride) 是第二代选择性且具有口服活性的雌激素受体 (estrogen receptor) 调节剂。Raloxifene hydrochloride 对骨脂代谢中，发挥雌激素激动作用，在子宫内膜和乳腺组织中具有雌激素拮抗作用。 |
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Sun, D., Jones, N.R., Manni, A., et al.Characterization of raloxifene glucuronidation: Potential role of UGT1A8 genotype on raloxifene metabolism in vivoCancer Prev. Res. (Phila.)6(7),719-730(2013)
Agency, W.A.-D.2014 Anti-doping testing figures report,(2014)
