Endoxifen E-isomer
Cat. No.:YN481642
产品名称: | Endoxifen E-isomer |
CAS No.: | 114828-90-9 |
Chemical Name: | 4-[(1E)-1-[4-[2-(methylamino)ethoxy]phenyl]-2-phenyl-1-buten-1-yl]phenol; E-Endoxifen |
Synonyms: | E-Endoxifen |
分子量: | 373.49 |
分子式: | C₂₅H₂₇NO₂ |
SMILES: | OC1=CC=C(/C(C2=CC=C(OCCNC)C=C2)=C(C3=CC=CC=C3)/CC)C=C1 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | Endoxifen E-isomer 是 (Z)-Endoxifen 的 E-异构体。(Z)-Endoxifen 是通过 CYP3A4/5 和 CYP2D6 作用产生的活性代谢物,是一种选择性雌激素受体调节剂 (SERM)。 |
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Furr, B., et al.: Pharmacol. Ther., 25, 127