Ezetimibe ketone
Cat. No.:YN410045
产品名称: | Ezetimibe ketone |
CAS No.: | 191330-56-0 |
Chemical Name: | (3R,4S)-1-(4-Fluorophenyl)-3-[3-(4-fluorophenyl)-3-oxopropyl]-4-(4-hydroxyphenyl)-2-azetidinone; EZM-K; Ezetimibe Ketone (USP) |
Synonyms: | EZM-K |
分子量: | 407.41 |
分子式: | C₂₄H₁₉F₂NO₃ |
SMILES: | O=C1N(C2=CC=C(F)C=C2)[C@H](C3=CC=C(O)C=C3)[C@H]1CCC(C4=CC=C(F)C=C4)=O |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | Ezetimibe ketone (EZM-K) 是 Ezetimibe 的 I 期代谢产物。Ezetimibe 是一种NPC1L1抑制剂,是有效的Nrf2激活剂,Ezetimibe 还是有效的胆固醇吸收抑制剂。 |
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Shah, V., et al: J. Pharm. Sci., 17, 1551 (2000),