Quisqualic acid
Cat. No.：YN320619
| 产品名称: | Quisqualic acid |
| CAS No.: | 52809-07-1 |
| Chemical Name: | αS-amino-3,5-dioxo-1,2,4-oxadiazolidine-2-propanoic acid |
| Synonyms: | |
| 分子量: | 189.13 |
| 分子式: | C₅H₇N₃O₅ |
| SMILES: | O=C(O)[C@@H](N)CN(C(N1)=O)OC1=O |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Quisqualic acid (L-Quisqualic acid) 是一种天然的谷氨酸类似物，是一种有效的，非选择性的兴奋性氨基酸 (EAA) 的两个亚型子集 (iGluR和mGluR) 激动剂，对 mGluR1R 的EC50为 45 nM，Kd值为 10 nM。Quisqualic acid 是从藜芦的果实中分离出来的。 |
| IC50和靶点: | [{name:"mGluR1R:45 nM (EC50)"},{name: "mGluR1R:10 nM (Ki)"},{name: "mGluR2R:108 μM (IC50)"},{name: "mGluR2R:113 μM (Ki)"},{name: "mGluR4R:593 μM (IC50)"},{name: "mGluR4R:112 μM (Ki)"}] |
| In Vitro: | |
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| Clinical Trial: | |
| Solvent & Solubility: |
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