VU0155041
Cat. No.:YN320864
CAS No. :1093757-42-6
产品名称: | VU0155041 |
CAS No.: | 1093757-42-6 |
Chemical Name: | |
Synonyms: | UV0155041,VU-0155041 |
分子量: | 316.18 |
分子式: | C₁₄H₁₅Cl₂NO₃ |
SMILES: | O=C([C@H](CCCC1)[C@H]1C(O)=O)NC2=CC(Cl)=CC(Cl)=C2 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | VU0155041 是一种有效,选择性的mGluR4混合变构激动剂/正变构调节剂 (PAM),对人和大鼠 mGluR4 的EC50值分别为 798 nM 和 693 nM。VU0155041 是 mGluR4 的部分激动剂,可通过与不同于谷氨酸结合位点的位点相互作用来激活受体。 |
IC50和靶点: | [{name:"Human mGlu4:798 nM (EC50)"},{name: "Rat mGlu4:693 nM (EC50)"}] |
In Vitro: | |
In Vivo: | |
Clinical Trial: | |
Solvent & Solubility: |