Ipatasertib dihydrochloride
Cat. No.：YN420201
CAS No. ：1396257-94-5
规格
价格(RMB)
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| 产品名称: | Ipatasertib dihydrochloride |
| CAS No.: | 1396257-94-5 |
| Chemical Name: | |
| Synonyms: | GDC-0068 dihydrochloride; RG-7440 dihydrochloride |
| 分子量: | 530.92 |
| 分子式: | C₂₄H₃₄Cl₃N₅O₂ |
| SMILES: | ClC1=CC=C([C@@H](CNC(C)C)C(N2CCN(C3=C([C@H](C)C[C@H]4O)C4=NC=N3)CC2)=O)C=C1.[H]Cl.[H]Cl |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Ipatasertib dihydrochloride (GDC-0068 dihydrochloride) 是一种选择性的，ATP竞争性的pan-Akt抑制剂，抑制Akt1，Akt2，Akt3的IC50分别为 5，18，8 nM。 |
| IC50和靶点: | [{name:"Akt1:5 nM (IC50)"},{name: "Akt3:8 nM (IC50)"},{name: "Akt2:18 nM (IC50)"},{name: "PKA:3100 nM (IC50)"}] |
| In Vitro: | |
| In Vivo: | |
| Clinical Trial: | |
| Solvent & Solubility: |
