FPA-124
Cat. No.：YN420212
CAS No. ：902779-59-3
规格
价格(RMB)
库存
| 产品名称: | FPA-124 |
| CAS No.: | 902779-59-3 |
| Chemical Name: | (SP-4-3)-dichloro[(2Z)-2-[(4-oxo-4H-1-benzopyran-3-yl)methylene]hydrazinecarbothioamide-κN2,κS]-copper |
| Synonyms: | |
| 分子量: | 381.73 |
| 分子式: | C₁₁H₉Cl₂CuN₃O₂S |
| SMILES: | O=C1C2=CC=CC=C2OC=C1/C=[N]3[Cu]([Cl-])([S]=C(N)N\3)[Cl-].[2+] |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | FPA-124，一种细胞通透性铜配合物，是选择性的Akt抑制剂，IC50为 0.1 μM ，与 Akt 的蛋白同源性 (PH) 域和激酶结构域相互作用。FPA-124 诱导细胞凋亡 (apoptosis)。 |
| IC50和靶点: | |
| In Vitro: | |
| In Vivo: | |
| Clinical Trial: | |
| Solvent & Solubility: |
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