Ligandrol
Cat. No.：YN481378
CAS No. ：1165910-22-4
规格
价格(RMB)
库存
| 产品名称: | Ligandrol |
| CAS No.: | 1165910-22-4 |
| Chemical Name: | 4-[(2R)-2-[(1R)-2,2,2-trifluoro-1-hydroxyethyl]-1-pyrrolidinyl]-2-(trifluoromethyl)-benzonitrile |
| Synonyms: | LGD-4033 |
| 分子量: | 338.25 |
| 分子式: | C₁₄H₁₂F₆N₂O |
| SMILES: | N#CC1=CC=C(N2[C@@H]([C@@H](O)C(F)(F)F)CCC2)C=C1C(F)(F)F |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Ligandrol (LGD-4033) 是一种新型的非类固醇，口服SARM，以高亲和力 (Ki为1 nM) 和选择性与雄激素受体结合。 |
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Basaria, S., Collins, L., Dillon, E.L., et al.The safety, pharmacokinetics, and effects of LGD-4033, a novel nonsteroidal oral, selective androgen receptor modulator, in healthy young menJ. Gerontol. A Biol. Sci. Med. Sci.68(1),87-95(2013)
Geldof, L., Pozo, O.J., Lootens, L., et al.In vitro metabolism study of a black market product containing SARM LGD-4033Drug Test Anal.9(2),168-178(2016)
Thevis, M., Lagojda, A., Kuehne, D., et al.Characterization of a non-approved selective androgen receptor modulator drug candidate sold via the internet and identification of in vitro generated phase-I metabolites for human sports drug testingRapid Commun Mass Spectrom.29(11),991-999(2015)
